Trial Outcomes & Findings for This Study is to Evaluate Safe and Effective Treatment Dose of OBI-888 in Patients With Locally Advanced or Metastatic Solid Tumors. (NCT NCT03573544)

NCT ID: NCT03573544

Last Updated: 2024-02-22

Results Overview

Assessment of OBI-888 clinical benefit rate for dose escalation and cohort expansion phases of the OBI-888-001 study.

Recruitment status

TERMINATED

Study phase

PHASE1/PHASE2

Target enrollment

54 participants

Primary outcome timeframe

Every 8 weeks (±1 week) for 6 months, then every 12 weeks (±1 week) until progression or off-study criteria, up to 1 year.

Results posted on

2024-02-22

Participant Flow

Participant milestones

Participant milestones
Measure
Part A, Dose Escalation - OBI-888 5 mg/kg
OBI-888 5 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part A, Dose Escalation - OBI-888 10 mg/kg
OBI-888 10 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part A, Dose Escalation - OBI-888 20 mg/kg
OBI-888 20 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part B, Cohort Expansion - Cohort 1, Pancreatic
OBI-888 20 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part B, Cohort Expansion - Cohort 2, Esophageal
OBI-888 20 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part B, Cohort Expansion - Cohort 3, Gastric
OBI-888 20 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part B, Cohort Expansion - Cohort 4, Colorectal
OBI-888 20 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part B, Cohort Expansion - Cohort 5, Basket
OBI-888 20 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Overall Study
STARTED
5
3
6
8
7
8
9
8
Overall Study
COMPLETED
0
0
0
0
0
0
0
0
Overall Study
NOT COMPLETED
5
3
6
8
7
8
9
8

Reasons for withdrawal

Reasons for withdrawal
Measure
Part A, Dose Escalation - OBI-888 5 mg/kg
OBI-888 5 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part A, Dose Escalation - OBI-888 10 mg/kg
OBI-888 10 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part A, Dose Escalation - OBI-888 20 mg/kg
OBI-888 20 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part B, Cohort Expansion - Cohort 1, Pancreatic
OBI-888 20 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part B, Cohort Expansion - Cohort 2, Esophageal
OBI-888 20 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part B, Cohort Expansion - Cohort 3, Gastric
OBI-888 20 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part B, Cohort Expansion - Cohort 4, Colorectal
OBI-888 20 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part B, Cohort Expansion - Cohort 5, Basket
OBI-888 20 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Overall Study
Adverse Event
0
0
0
3
1
0
2
0
Overall Study
Physician Decision
0
0
0
0
0
0
1
0
Overall Study
Withdrawal by Subject
2
0
0
1
1
1
0
1
Overall Study
Disease progression
3
3
6
4
5
7
6
7

Baseline Characteristics

This Study is to Evaluate Safe and Effective Treatment Dose of OBI-888 in Patients With Locally Advanced or Metastatic Solid Tumors.

Baseline characteristics by cohort

Baseline characteristics by cohort
Measure
Part A, Dose Escalation - OBI-888 5 mg/kg
n=5 Participants
OBI-888 5 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part A, Dose Escalation - OBI-888 10 mg/kg
n=3 Participants
OBI-888 10 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part A, Dose Escalation - OBI-888 20 mg/kg
n=6 Participants
OBI-888 20 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part B, Cohort Expansion - Cohort 1, Pancreatic
n=8 Participants
OBI-888 20 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part B, Cohort Expansion - Cohort 2, Esophageal
n=7 Participants
OBI-888 20 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part B, Cohort Expansion - Cohort 3, Gastric
n=8 Participants
OBI-888 20 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part B, Cohort Expansion - Cohort 4, Colorectal
n=9 Participants
OBI-888 20 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part B, Cohort Expansion - Cohort 5, Basket
n=8 Participants
OBI-888 20 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Total
n=54 Participants
Total of all reporting groups
Age, Continuous
51 years
STANDARD_DEVIATION 12.86 • n=99 Participants
57.7 years
STANDARD_DEVIATION 9.45 • n=107 Participants
64.5 years
STANDARD_DEVIATION 12.1 • n=206 Participants
63.8 years
STANDARD_DEVIATION 13.29 • n=157 Participants
57.4 years
STANDARD_DEVIATION 9.36 • n=390 Participants
64.9 years
STANDARD_DEVIATION 9.69 • n=16 Participants
52.9 years
STANDARD_DEVIATION 14.84 • n=3 Participants
60.6 years
STANDARD_DEVIATION 8.07 • n=6 Participants
59.8 years
STANDARD_DEVIATION 11.81 • n=114 Participants
Sex: Female, Male
Female
5 Participants
n=99 Participants
3 Participants
n=107 Participants
3 Participants
n=206 Participants
6 Participants
n=157 Participants
0 Participants
n=390 Participants
3 Participants
n=16 Participants
2 Participants
n=3 Participants
5 Participants
n=6 Participants
27 Participants
n=114 Participants
Sex: Female, Male
Male
0 Participants
n=99 Participants
0 Participants
n=107 Participants
3 Participants
n=206 Participants
2 Participants
n=157 Participants
7 Participants
n=390 Participants
5 Participants
n=16 Participants
7 Participants
n=3 Participants
3 Participants
n=6 Participants
27 Participants
n=114 Participants
Race (NIH/OMB)
American Indian or Alaska Native
0 Participants
n=99 Participants
0 Participants
n=107 Participants
0 Participants
n=206 Participants
0 Participants
n=157 Participants
0 Participants
n=390 Participants
0 Participants
n=16 Participants
0 Participants
n=3 Participants
0 Participants
n=6 Participants
0 Participants
n=114 Participants
Race (NIH/OMB)
Asian
0 Participants
n=99 Participants
0 Participants
n=107 Participants
1 Participants
n=206 Participants
3 Participants
n=157 Participants
6 Participants
n=390 Participants
7 Participants
n=16 Participants
0 Participants
n=3 Participants
4 Participants
n=6 Participants
21 Participants
n=114 Participants
Race (NIH/OMB)
Native Hawaiian or Other Pacific Islander
0 Participants
n=99 Participants
0 Participants
n=107 Participants
0 Participants
n=206 Participants
0 Participants
n=157 Participants
0 Participants
n=390 Participants
0 Participants
n=16 Participants
0 Participants
n=3 Participants
0 Participants
n=6 Participants
0 Participants
n=114 Participants
Race (NIH/OMB)
Black or African American
1 Participants
n=99 Participants
1 Participants
n=107 Participants
0 Participants
n=206 Participants
0 Participants
n=157 Participants
0 Participants
n=390 Participants
0 Participants
n=16 Participants
0 Participants
n=3 Participants
0 Participants
n=6 Participants
2 Participants
n=114 Participants
Race (NIH/OMB)
White
3 Participants
n=99 Participants
1 Participants
n=107 Participants
5 Participants
n=206 Participants
5 Participants
n=157 Participants
1 Participants
n=390 Participants
1 Participants
n=16 Participants
9 Participants
n=3 Participants
4 Participants
n=6 Participants
29 Participants
n=114 Participants
Race (NIH/OMB)
More than one race
0 Participants
n=99 Participants
0 Participants
n=107 Participants
0 Participants
n=206 Participants
0 Participants
n=157 Participants
0 Participants
n=390 Participants
0 Participants
n=16 Participants
0 Participants
n=3 Participants
0 Participants
n=6 Participants
0 Participants
n=114 Participants
Race (NIH/OMB)
Unknown or Not Reported
1 Participants
n=99 Participants
1 Participants
n=107 Participants
0 Participants
n=206 Participants
0 Participants
n=157 Participants
0 Participants
n=390 Participants
0 Participants
n=16 Participants
0 Participants
n=3 Participants
0 Participants
n=6 Participants
2 Participants
n=114 Participants
Race/Ethnicity, Customized
Ethnicity (NIH/OMB) · Hispanic or Latino
1 Participants
n=99 Participants
0 Participants
n=107 Participants
1 Participants
n=206 Participants
0 Participants
n=157 Participants
0 Participants
n=390 Participants
0 Participants
n=16 Participants
0 Participants
n=3 Participants
0 Participants
n=6 Participants
2 Participants
n=114 Participants
Race/Ethnicity, Customized
Ethnicity (NIH/OMB) · Not Hispanic or Latino
0 Participants
n=99 Participants
0 Participants
n=107 Participants
0 Participants
n=206 Participants
0 Participants
n=157 Participants
0 Participants
n=390 Participants
0 Participants
n=16 Participants
0 Participants
n=3 Participants
0 Participants
n=6 Participants
0 Participants
n=114 Participants
Race/Ethnicity, Customized
Ethnicity (NIH/OMB) · East Asian
0 Participants
n=99 Participants
0 Participants
n=107 Participants
0 Participants
n=206 Participants
3 Participants
n=157 Participants
6 Participants
n=390 Participants
7 Participants
n=16 Participants
0 Participants
n=3 Participants
3 Participants
n=6 Participants
19 Participants
n=114 Participants
Race/Ethnicity, Customized
Ethnicity (NIH/OMB) · Other
2 Participants
n=99 Participants
2 Participants
n=107 Participants
3 Participants
n=206 Participants
4 Participants
n=157 Participants
1 Participants
n=390 Participants
1 Participants
n=16 Participants
8 Participants
n=3 Participants
3 Participants
n=6 Participants
24 Participants
n=114 Participants
Race/Ethnicity, Customized
Ethnicity (NIH/OMB) · Unknown or not reported
2 Participants
n=99 Participants
1 Participants
n=107 Participants
2 Participants
n=206 Participants
1 Participants
n=157 Participants
0 Participants
n=390 Participants
0 Participants
n=16 Participants
1 Participants
n=3 Participants
2 Participants
n=6 Participants
9 Participants
n=114 Participants

PRIMARY outcome

Timeframe: Every 8 weeks (±1 week) for 6 months, then every 12 weeks (±1 week) until progression or off-study criteria, up to 1 year.

Assessment of OBI-888 clinical benefit rate for dose escalation and cohort expansion phases of the OBI-888-001 study.

Outcome measures

Outcome measures
Measure
Part A, Dose Escalation - OBI-888 5 mg/kg
n=5 Participants
OBI-888 5 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part A, Dose Escalation - OBI-888 10 mg/kg
n=3 Participants
OBI-888 10 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part A, Dose Escalation - OBI-888 20 mg/kg
n=6 Participants
OBI-888 20 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part B, Cohort Expansion - Cohort 1, Pancreatic
n=8 Participants
OBI-888 20 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part B, Cohort Expansion - Cohort 2, Esophageal
n=7 Participants
OBI-888 20 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part B, Cohort Expansion - Cohort 3, Gastric
n=8 Participants
OBI-888 20 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part B, Cohort Expansion - Cohort 4, Colorectal
n=9 Participants
OBI-888 20 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part B, Cohort Expansion - Cohort 5, Basket
n=8 Participants
OBI-888 20 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Clinical Benefit Rate (CR, PR, SD) (%)
20 Percentage
Interval 0.5 to 71.6
66.7 Percentage
Interval 9.4 to 99.2
16.7 Percentage
Interval 0.4 to 64.1
12.5 Percentage
Interval 0.3 to 52.7
14.3 Percentage
Interval 0.4 to 57.9
25 Percentage
Interval 3.2 to 65.1
22.2 Percentage
Interval 2.8 to 60.0
25 Percentage
Interval 3.2 to 65.1

Adverse Events

Part A, Dose Escalation - OBI-888 5 mg/kg

Serious events: 1 serious events
Other events: 5 other events
Deaths: 0 deaths

Part A, Dose Escalation - OBI-888 10 mg/kg

Serious events: 1 serious events
Other events: 3 other events
Deaths: 0 deaths

Part A, Dose Escalation - OBI-888 20 mg/kg

Serious events: 0 serious events
Other events: 5 other events
Deaths: 0 deaths

Part B, Cohort Expansion - Cohort 1, Pancreatic

Serious events: 8 serious events
Other events: 8 other events
Deaths: 1 deaths

Part B, Cohort Expansion - Cohort 2, Esophageal

Serious events: 2 serious events
Other events: 6 other events
Deaths: 0 deaths

Part B, Cohort Expansion - Cohort 3, Gastric

Serious events: 5 serious events
Other events: 8 other events
Deaths: 0 deaths

Part B, Cohort Expansion - Cohort 4, Colorectal

Serious events: 5 serious events
Other events: 9 other events
Deaths: 1 deaths

Part B, Cohort Expansion - Cohort 5, Basket

Serious events: 2 serious events
Other events: 8 other events
Deaths: 0 deaths

Serious adverse events

Serious adverse events
Measure
Part A, Dose Escalation - OBI-888 5 mg/kg
n=5 participants at risk
OBI-888 5 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part A, Dose Escalation - OBI-888 10 mg/kg
n=3 participants at risk
OBI-888 10 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part A, Dose Escalation - OBI-888 20 mg/kg
n=6 participants at risk
OBI-888 20 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part B, Cohort Expansion - Cohort 1, Pancreatic
n=8 participants at risk
OBI-888 20 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part B, Cohort Expansion - Cohort 2, Esophageal
n=7 participants at risk
OBI-888 20 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part B, Cohort Expansion - Cohort 3, Gastric
n=8 participants at risk
OBI-888 20 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part B, Cohort Expansion - Cohort 4, Colorectal
n=9 participants at risk
OBI-888 20 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part B, Cohort Expansion - Cohort 5, Basket
n=8 participants at risk
OBI-888 20 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Blood and lymphatic system disorders
Anaemia
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Cardiac disorders
Supraventricular tachycardia
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
11.1%
1/9 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Gastrointestinal disorders
Abdominal pain
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
11.1%
1/9 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Gastrointestinal disorders
Gastric ulcer
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
11.1%
1/9 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Gastrointestinal disorders
Gastrointestinal haemorrhage
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
25.0%
2/8 • Number of events 3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Gastrointestinal disorders
Haematemesis
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
14.3%
1/7 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Gastrointestinal disorders
Intestinal obstruction
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 2 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Gastrointestinal disorders
Nausea
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Gastrointestinal disorders
Oesophageal rupture
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
14.3%
1/7 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Gastrointestinal disorders
Upper gastrointestinal haemorrhage
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Gastrointestinal disorders
Vomiting
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
11.1%
1/9 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
General disorders
Fatigue
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Hepatobiliary disorders
Cholangitis
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Hepatobiliary disorders
Jaundice
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Infections and infestations
Bacteremia
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Infections and infestations
Biliary tract infection
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Infections and infestations
Cellulitis
20.0%
1/5 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Infections and infestations
Pneumonia
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Infections and infestations
Sepsis
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Injury, poisoning and procedural complications
Fall
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Injury, poisoning and procedural complications
Infusion related reaction
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Investigations
Blood bilirubin increased
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Investigations
Blood creatinine increased
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Metabolism and nutrition disorders
Failure to thrive
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Musculoskeletal and connective tissue disorders
Muscular weakness
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Psychiatric disorders
Mental status changes
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Renal and urinary disorders
Hydronephrosis
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Renal and urinary disorders
Acute kidney injury
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
25.0%
2/8 • Number of events 2 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Renal and urinary disorders
Renal failure
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
11.1%
1/9 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Respiratory, thoracic and mediastinal disorders
Pleural effusion
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
33.3%
1/3 • Number of events 2 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Vascular disorders
Shock
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B

Other adverse events

Other adverse events
Measure
Part A, Dose Escalation - OBI-888 5 mg/kg
n=5 participants at risk
OBI-888 5 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part A, Dose Escalation - OBI-888 10 mg/kg
n=3 participants at risk
OBI-888 10 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part A, Dose Escalation - OBI-888 20 mg/kg
n=6 participants at risk
OBI-888 20 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part B, Cohort Expansion - Cohort 1, Pancreatic
n=8 participants at risk
OBI-888 20 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part B, Cohort Expansion - Cohort 2, Esophageal
n=7 participants at risk
OBI-888 20 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part B, Cohort Expansion - Cohort 3, Gastric
n=8 participants at risk
OBI-888 20 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part B, Cohort Expansion - Cohort 4, Colorectal
n=9 participants at risk
OBI-888 20 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Part B, Cohort Expansion - Cohort 5, Basket
n=8 participants at risk
OBI-888 20 mg/kg was administered as an IV infusion for approximately 90 minutes (±10 minutes) on Days 1, 8, 15 and 22 of each 28-day cycle for 2 cycles
Gastrointestinal disorders
Vomiting
40.0%
2/5 • Number of events 2 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
14.3%
1/7 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
37.5%
3/8 • Number of events 3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
33.3%
3/9 • Number of events 6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
25.0%
2/8 • Number of events 3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Gastrointestinal disorders
Nausea
40.0%
2/5 • Number of events 2 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
16.7%
1/6 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
25.0%
2/8 • Number of events 3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
37.5%
3/8 • Number of events 3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
11.1%
1/9 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 2 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Gastrointestinal disorders
Abdominal pain
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
33.3%
2/6 • Number of events 2 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
25.0%
2/8 • Number of events 6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
14.3%
1/7 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
22.2%
2/9 • Number of events 2 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
37.5%
3/8 • Number of events 3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Gastrointestinal disorders
Constipation
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
16.7%
1/6 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
25.0%
2/8 • Number of events 2 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
25.0%
2/8 • Number of events 2 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
11.1%
1/9 • Number of events 2 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Gastrointestinal disorders
Diarrhoea
20.0%
1/5 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
14.3%
1/7 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
11.1%
1/9 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
37.5%
3/8 • Number of events 3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
General disorders
Fatigue
40.0%
2/5 • Number of events 2 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
33.3%
1/3 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
33.3%
2/6 • Number of events 2 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
50.0%
4/8 • Number of events 4 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
28.6%
2/7 • Number of events 2 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
50.0%
4/8 • Number of events 4 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
22.2%
2/9 • Number of events 3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
37.5%
3/8 • Number of events 4 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
General disorders
Pyrexia
40.0%
2/5 • Number of events 3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
37.5%
3/8 • Number of events 5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
General disorders
Chills
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
25.0%
2/8 • Number of events 2 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
14.3%
1/7 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
22.2%
2/9 • Number of events 2 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
25.0%
2/8 • Number of events 2 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
General disorders
Asthenia
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
16.7%
1/6 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
25.0%
2/8 • Number of events 2 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
25.0%
2/8 • Number of events 2 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
General disorders
Oedema peripheral
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
16.7%
1/6 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
General disorders
Peripheral swelling
20.0%
1/5 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
14.3%
1/7 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Metabolism and nutrition disorders
Decreased appetite
60.0%
3/5 • Number of events 3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
16.7%
1/6 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
37.5%
3/8 • Number of events 3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
11.1%
1/9 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Metabolism and nutrition disorders
Hyperkalaemia
20.0%
1/5 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
16.7%
1/6 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
37.5%
3/8 • Number of events 3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Metabolism and nutrition disorders
Hypokalaemia
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
16.7%
1/6 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
25.0%
2/8 • Number of events 2 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Metabolism and nutrition disorders
Hyponatremia
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
25.0%
2/8 • Number of events 2 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Respiratory, thoracic and mediastinal disorders
Dyspnoea
40.0%
2/5 • Number of events 4 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
50.0%
3/6 • Number of events 3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
14.3%
1/7 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 2 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Respiratory, thoracic and mediastinal disorders
Pleural effusion
20.0%
1/5 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
33.3%
1/3 • Number of events 2 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
16.7%
1/6 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
14.3%
1/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Respiratory, thoracic and mediastinal disorders
Cough
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
14.3%
1/7 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
25.0%
2/8 • Number of events 3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Musculoskeletal and connective tissue disorders
Back pain
20.0%
1/5 • Number of events 2 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
22.2%
2/9 • Number of events 2 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
25.0%
2/8 • Number of events 2 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Musculoskeletal and connective tissue disorders
Arthralgia
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
33.3%
1/3 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
16.7%
1/6 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Musculoskeletal and connective tissue disorders
Muscular weakness
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
14.3%
1/7 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Investigations
Aspartate aminotransferase increased
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
25.0%
2/8 • Number of events 2 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
37.5%
3/8 • Number of events 6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Investigations
Blood creatinine increased
20.0%
1/5 • Number of events 2 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
16.7%
1/6 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
11.1%
1/9 • Number of events 3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Investigations
Blood bilirubin increased
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
11.1%
1/9 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
25.0%
2/8 • Number of events 2 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Blood and lymphatic system disorders
Anaemia
40.0%
2/5 • Number of events 2 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
33.3%
1/3 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
28.6%
2/7 • Number of events 2 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
25.0%
2/8 • Number of events 8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
22.2%
2/9 • Number of events 4 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Blood and lymphatic system disorders
Leukocytosis
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
22.2%
2/9 • Number of events 2 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Nervous system disorders
Headache
60.0%
3/5 • Number of events 3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
11.1%
1/9 • Number of events 2 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Nervous system disorders
Dizziness
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
16.7%
1/6 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
25.0%
2/8 • Number of events 2 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Renal and urinary disorders
Acute kidney injury
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/9 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
25.0%
2/8 • Number of events 2 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Renal and urinary disorders
Hydronephrosis
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
25.0%
2/8 • Number of events 2 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
11.1%
1/9 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Renal and urinary disorders
Renal failure
20.0%
1/5 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/3 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
11.1%
1/9 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
Injury, poisoning and procedural complications
Infusion related reaction
0.00%
0/5 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
33.3%
1/3 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/6 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/7 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
12.5%
1/8 • Number of events 1 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
22.2%
2/9 • Number of events 4 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B
0.00%
0/8 • Adverse event data were collected through 12 months
Treatment-emergent adverse events (TEAEs) in Parts A or B experienced by ≥5% of total subjects in Part A and Part B. TEAEs are presented by decreasing incidence for the total of subjects in Part A and Part B

Additional Information

Dr. Wayne Saville, Chief Medical Officer

OBI Pharma, Inc.

Phone: 619-537-7821

Results disclosure agreements

  • Principal investigator is a sponsor employee
  • Publication restrictions are in place