Trial Outcomes & Findings for A Study of LY2409021 in Healthy Participants (NCT NCT02217618)

NCT ID: NCT02217618

Last Updated: 2018-10-29

Results Overview

Area under the concentration versus time curve from zero to infinity (AUC\[0-inf\]) of LY2409021 is presented.

Recruitment status

COMPLETED

Study phase

PHASE1

Target enrollment

16 participants

Primary outcome timeframe

Pre-dose and 0.5, 1, 2, 4, 8, 12, 24, 48, 72, 96, 144, 192, 264, and 336 hours post-dose

Results posted on

2018-10-29

Participant Flow

Participant milestones

Participant milestones
Measure
LY2409021
Single oral dose of 20 milligrams (mg) LY2409021.
Overall Study
STARTED
16
Overall Study
Received Study Drug
16
Overall Study
COMPLETED
16
Overall Study
NOT COMPLETED
0

Reasons for withdrawal

Withdrawal data not reported

Baseline Characteristics

A Study of LY2409021 in Healthy Participants

Baseline characteristics by cohort

Baseline characteristics by cohort
Measure
LY2409021
n=16 Participants
Single oral dose of 20 mg LY2409021.
Age, Continuous
48.4 years
STANDARD_DEVIATION 13.3 • n=99 Participants
Sex: Female, Male
Female
7 Participants
n=99 Participants
Sex: Female, Male
Male
9 Participants
n=99 Participants
Ethnicity (NIH/OMB)
Hispanic or Latino
2 Participants
n=99 Participants
Ethnicity (NIH/OMB)
Not Hispanic or Latino
14 Participants
n=99 Participants
Ethnicity (NIH/OMB)
Unknown or Not Reported
0 Participants
n=99 Participants
Race (NIH/OMB)
American Indian or Alaska Native
0 Participants
n=99 Participants
Race (NIH/OMB)
Asian
0 Participants
n=99 Participants
Race (NIH/OMB)
Native Hawaiian or Other Pacific Islander
0 Participants
n=99 Participants
Race (NIH/OMB)
Black or African American
2 Participants
n=99 Participants
Race (NIH/OMB)
White
14 Participants
n=99 Participants
Race (NIH/OMB)
More than one race
0 Participants
n=99 Participants
Race (NIH/OMB)
Unknown or Not Reported
0 Participants
n=99 Participants
Region of Enrollment
United States
16 Participants
n=99 Participants

PRIMARY outcome

Timeframe: Pre-dose and 0.5, 1, 2, 4, 8, 12, 24, 48, 72, 96, 144, 192, 264, and 336 hours post-dose

Population: All participants who received a dose of study drug and had evaluable AUC(0-inf) data.

Area under the concentration versus time curve from zero to infinity (AUC\[0-inf\]) of LY2409021 is presented.

Outcome measures

Outcome measures
Measure
LY2409021
n=16 Participants
Single oral dose of 20 mg LY2409021.
Pharmacokinetics: Area Under the Concentration Curve (AUC) of LY2409021
48100 nanogram*hours per milliliter (ng*h/mL)
Geometric Coefficient of Variation 28

PRIMARY outcome

Timeframe: Pre-dose and 0.5, 1, 2, 4, 8, 12, 24, 48, 72, 96, 144, 192, 264, and 336 hours post-dose

Population: All participants who received a dose of study drug and had evaluable Cmax data.

Outcome measures

Outcome measures
Measure
LY2409021
n=16 Participants
Single oral dose of 20 mg LY2409021.
Pharmacokinetics: Maximum Concentration (Cmax) of LY2409021
625 nanograms per milliliter (ng/mL)
Geometric Coefficient of Variation 29

PRIMARY outcome

Timeframe: Pre-dose and 0.5, 1, 2, 4, 8, 12, 24, 48, 72, 96, 144, 192, 264, and 336 hours post-dose

Population: All participants who received a dose of study drug and had evaluable Tmax data.

Outcome measures

Outcome measures
Measure
LY2409021
n=16 Participants
Single oral dose of 20 mg LY2409021.
Pharmacokinetics: Time to Maximum Observed Drug Concentration (Tmax) of LY2409021
8.00 hours
Interval 4.0 to 24.03

Adverse Events

LY2409021

Serious events: 0 serious events
Other events: 3 other events
Deaths: 0 deaths

Serious adverse events

Adverse event data not reported

Other adverse events

Other adverse events
Measure
LY2409021
n=16 participants at risk
Single oral dose of 20 mg LY2409021.
Gastrointestinal disorders
Abdominal pain
6.2%
1/16 • Number of events 1
Nervous system disorders
Headache
6.2%
1/16 • Number of events 1
Skin and subcutaneous tissue disorders
Miliaria
6.2%
1/16 • Number of events 1

Additional Information

Chief Medical Officer

Eli Lilly and Company

Phone: 800-545-5979

Results disclosure agreements

  • Principal investigator is a sponsor employee
  • Publication restrictions are in place

Restriction type: GT60