Trial Outcomes & Findings for Long-term Efficacy, Safety and Tolerability of Pramipexole in Patients With Idiopathic Moderate to Severe Restless Legs Syndrome (RLS) (NCT NCT00472199)

NCT ID: NCT00472199

Last Updated: 2014-06-27

Results Overview

IRLS total score ranging from 0 (no RLS symptoms) to 40 (very severe RLS symptoms)

Recruitment status

COMPLETED

Study phase

PHASE4

Target enrollment

331 participants

Primary outcome timeframe

Baseline and 26 weeks

Results posted on

2014-06-27

Participant Flow

Of 331 patients enrolled, 329 were treated with study drug. Two patients were randomized, but before their first intake of trial medication they decided to not participate in the study.

Participant milestones

Participant milestones
Measure
Pramipexole
4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase the dose to 0.25mg and to further increase or decrease the dose in steps to 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Placebo
4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Overall Study
STARTED
166
163
Overall Study
COMPLETED
131
103
Overall Study
NOT COMPLETED
35
60

Reasons for withdrawal

Reasons for withdrawal
Measure
Pramipexole
4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase the dose to 0.25mg and to further increase or decrease the dose in steps to 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Placebo
4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Overall Study
Adverse Event
19
23
Overall Study
Lack of Efficacy
4
25
Overall Study
Lost to Follow-up
2
4
Overall Study
Protocol Violation
3
2
Overall Study
Withdrawal by Subject
6
5
Overall Study
personal reason
0
1
Overall Study
patient was asymptomatic
1
0

Baseline Characteristics

Long-term Efficacy, Safety and Tolerability of Pramipexole in Patients With Idiopathic Moderate to Severe Restless Legs Syndrome (RLS)

Baseline characteristics by cohort

Baseline characteristics by cohort
Measure
Pramipexole
n=166 Participants
4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase the dose to 0.25mg and to further increase or decrease the dose in steps to 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Placebo
n=163 Participants
4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Total
n=329 Participants
Total of all reporting groups
Age, Continuous
57.9 years
STANDARD_DEVIATION 12.7 • n=99 Participants
55.8 years
STANDARD_DEVIATION 11.4 • n=107 Participants
56.8 years
STANDARD_DEVIATION 12.1 • n=206 Participants
Sex: Female, Male
Female
102 Participants
n=99 Participants
94 Participants
n=107 Participants
196 Participants
n=206 Participants
Sex: Female, Male
Male
64 Participants
n=99 Participants
69 Participants
n=107 Participants
133 Participants
n=206 Participants

PRIMARY outcome

Timeframe: Baseline and 26 weeks

Population: Intent to treat analysis. Number of randomized patients with a baseline and at least one non-missing post-baseline measure. Imputation by last observation carried forward (LOCF) for post-baseline values

IRLS total score ranging from 0 (no RLS symptoms) to 40 (very severe RLS symptoms)

Outcome measures

Outcome measures
Measure
Pramipexole
n=162 Participants
4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase the dose to 0.25mg and to further increase or decrease the dose in steps to 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Placebo
n=159 Participants
4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Change From Baseline in International Restless Legs Syndrome Study Group Rating Scale (IRLS) Total Score After 26 Weeks
-13.7 Scores on a scale
Standard Error 0.8
-11.1 Scores on a scale
Standard Error 0.8

SECONDARY outcome

Timeframe: after 26 weeks of treatment

Population: Intent to treat analysis. Number of randomized patients with a baseline and at least one non-missing post-baseline measure. Imputation by last observation carried forward (LOCF) for post-baseline values.

CGI-I scores ranging from '1' (very much improved) to '7' (very much worse), CGI-I responder have scoring 1 or 2 (at least much improved)

Outcome measures

Outcome measures
Measure
Pramipexole
n=162 Participants
4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase the dose to 0.25mg and to further increase or decrease the dose in steps to 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Placebo
n=159 Participants
4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Clinical Global Impression - Global Improvement (CGI-I) Responder Rate
CGI-I responder (at least much improved)
111 participants
80 participants
Clinical Global Impression - Global Improvement (CGI-I) Responder Rate
CGI-I non-responder
51 participants
79 participants

SECONDARY outcome

Timeframe: after 26 weeks of treatment

Population: Intent to treat analysis. Number of randomized patients with a baseline and at least one non-missing post-baseline measure. Imputation by last observation carried forward (LOCF) for post-baseline values

IRLS response was defined as at least 50% reduction in IRLS total score from baseline. IRLS total score ranging from 0 (no RLS symptoms) to 40 (very severe symptoms)

Outcome measures

Outcome measures
Measure
Pramipexole
n=162 Participants
4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase the dose to 0.25mg and to further increase or decrease the dose in steps to 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Placebo
n=159 Participants
4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
International Restless Legs Syndrome (IRLS) Study Group Rating Scale Responder Rate
IRLS responder
95 participants
68 participants
International Restless Legs Syndrome (IRLS) Study Group Rating Scale Responder Rate
IRLS non-responder
67 participants
91 participants

SECONDARY outcome

Timeframe: after 26 weeks of treatment

Population: Intent to treat analysis. Number of randomized patients with a baseline and at least one non-missing post-baseline measure. Imputation by last observation carried forward (LOCF) for post-baseline values

PGI scores ranging from '1' (very much better) to '7' (very much worse), PGI responder have scoring 1 or 2 (at least much better)

Outcome measures

Outcome measures
Measure
Pramipexole
n=162 Participants
4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase the dose to 0.25mg and to further increase or decrease the dose in steps to 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Placebo
n=159 Participants
4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Patient Global Impression (PGI) Responder Rate
PGI responder (much better or very much better)
101 participants
70 participants
Patient Global Impression (PGI) Responder Rate
PGI non-responder
61 participants
89 participants

SECONDARY outcome

Timeframe: baseline and 26 weeks of treatment

Population: Intent to treat analysis. Number of randomized patients with a baseline and at least one non-missing post-baseline measure. Imputation by last observation carried forward (LOCF) for post-baseline values

The score is an 11-point Likert scale, ranging from "none/not at all" (0) to "very severe" (10), to reflect the patient's condition during the previous week

Outcome measures

Outcome measures
Measure
Pramipexole
n=162 Participants
4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase the dose to 0.25mg and to further increase or decrease the dose in steps to 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Placebo
n=159 Participants
4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Change From Baseline in Restless Legs Syndrome-6 (RLS-6) Score "Satisfaction With Sleep" After 26 Weeks
-2.5 Scores on a scale
Interval -5.0 to 0.0
-2 Scores on a scale
Interval -4.0 to 0.0

SECONDARY outcome

Timeframe: Baseline and 26 weeks of treatment

Population: Intent to treat analysis. Number of randomized patients with a baseline and at least one non-missing post-baseline measure. Imputation by last observation carried forward (LOCF) for post-baseline values

The score is an 11-point Likert scale, ranging from "none/not at all" (0) to "very severe" (10), to reflect the patient's condition during the previous week

Outcome measures

Outcome measures
Measure
Pramipexole
n=162 Participants
4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase the dose to 0.25mg and to further increase or decrease the dose in steps to 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Placebo
n=159 Participants
4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Change From Baseline in RLS-6 Score "Severity Falling Asleep" After 26 Weeks
-3 Scores on a scale
Interval -5.0 to 0.0
-1 Scores on a scale
Interval -4.0 to 0.0

SECONDARY outcome

Timeframe: baseline and 26 weeks of treatment

Population: Intent to treat analysis. Number of randomized patients with a baseline and at least one non-missing post-baseline measure. Imputation by last observation carried forward (LOCF) for post-baseline values

The question was rated on an 11-point Likert scale, ranging from "none/not at all" (0) to "very severe" (10), to reflect the patient's condition during the previous week

Outcome measures

Outcome measures
Measure
Pramipexole
n=162 Participants
4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase the dose to 0.25mg and to further increase or decrease the dose in steps to 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Placebo
n=159 Participants
4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Change From Baseline in RLS-6 Score "Severity During the Night" After 26 Weeks
-3 Scores on a scale
Interval -5.0 to 0.0
-2 Scores on a scale
Interval -5.0 to 0.0

SECONDARY outcome

Timeframe: Baseline and 26 weeks of treatment

Population: Intent to treat analysis. Number of randomized patients with a baseline and at least one non-missing post-baseline measure. Imputation by last observation carried forward (LOCF) for post-baseline values

The score is an 11-point Likert scale, ranging from "none/not at all" (0) to "very severe" (10), to reflect the patient's condition during the previous week

Outcome measures

Outcome measures
Measure
Pramipexole
n=162 Participants
4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase the dose to 0.25mg and to further increase or decrease the dose in steps to 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Placebo
n=159 Participants
4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Change From Baseline in RLS-6 Score "Severity During the Day When at Rest" After 26 Weeks
-3 Scores on a scale
Interval -5.0 to 0.0
-1 Scores on a scale
Interval -4.0 to 0.0

SECONDARY outcome

Timeframe: Baseline and 26 weeks of treatment

Population: Intent to treat analysis. Number of randomized patients with a baseline and at least one non-missing post-baseline measure. Imputation by last observation carried forward (LOCF) for post-baseline values

The score is an 11-point Likert scale, ranging from "none/not at all" (0) to "very severe" (10), to reflect the patient's condition during the previous week

Outcome measures

Outcome measures
Measure
Pramipexole
n=162 Participants
4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase the dose to 0.25mg and to further increase or decrease the dose in steps to 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Placebo
n=159 Participants
4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Change From Baseline RLS-6 Score "Severity During the Day Engaged in Activities" After 26 Weeks
0 Scores on a scale
Interval -1.0 to 0.0
0 Scores on a scale
Interval -1.0 to 0.0

SECONDARY outcome

Timeframe: Baseline and 26 weeks of treatment

Population: Intent to treat analysis. Number of randomized patients with a baseline and at least one non-missing post-baseline measure. Imputation by last observation carried forward (LOCF) for post-baseline values

The score is an 11-point Likert scale, ranging from "none/not at all" (0) to "very severe" (10), to reflect the patient's condition during the previous week

Outcome measures

Outcome measures
Measure
Pramipexole
n=162 Participants
4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase the dose to 0.25mg and to further increase or decrease the dose in steps to 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Placebo
n=159 Participants
4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Change From Baseline in RLS-6 Score "Tired or Sleepy During the Day" After 26 Weeks
-1 Scores on a scale
Interval -3.0 to 0.0
-1 Scores on a scale
Interval -3.0 to 0.0

SECONDARY outcome

Timeframe: Baseline and 26 weeks of treatment

Population: Intent to treat analysis. Number of randomized patients with a baseline and at least one non-missing post-baseline measure. Imputation by last observation carried forward (LOCF) for post-baseline values

Mood disturbance associated with RLS symptoms ranging from 0 (none) to 4 (very severe)

Outcome measures

Outcome measures
Measure
Pramipexole
n=162 Participants
4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase the dose to 0.25mg and to further increase or decrease the dose in steps to 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Placebo
n=159 Participants
4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Change From Baseline in IRLS Mood Disturbance Score (Item 10) After 26 Weeks
-1 scores on a scale
Interval -2.0 to 0.0
-1 scores on a scale
Interval -2.0 to 0.0

SECONDARY outcome

Timeframe: Baseline and 26 weeks of treatment

Population: Intent to treat analysis. Number of randomized patients with a baseline and at least one non-missing post-baseline measure. Imputation by last observation carried forward (LOCF) for post-baseline values

The scale measures pain on a continuous 100 mm axis ranging from no pain (0 mm) to unbearable pain (100 mm)

Outcome measures

Outcome measures
Measure
Pramipexole
n=162 Participants
4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase the dose to 0.25mg and to further increase or decrease the dose in steps to 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Placebo
n=158 Participants
4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Change From Baseline in Visual Analogue Scale (VAS) Score for Pain in Limbs After 26 Weeks
-26 Scores on a scale
Interval -47.0 to -5.0
-15 Scores on a scale
Interval -46.0 to 0.0

SECONDARY outcome

Timeframe: Baseline and 26 weeks of treatment

Population: Intent to treat analysis. Number of randomized patients with a baseline and at least one non-missing post-baseline measure. Imputation by last observation carried forward (LOCF) for post-baseline values

RLS QoL total score ranging from 0 to 100 with higher values indicating better quality of life

Outcome measures

Outcome measures
Measure
Pramipexole
n=157 Participants
4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase the dose to 0.25mg and to further increase or decrease the dose in steps to 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Placebo
n=153 Participants
4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Change From Baseline in Quality of Life in RLS (RLS QoL) Score After 26 Weeks
15 Scores on a scale
Interval 5.0 to 25.0
12.5 Scores on a scale
Interval 2.5 to 27.5

SECONDARY outcome

Timeframe: Baseline and 26 weeks

Population: Intent to treat analysis. Number of randomized patients with a baseline and at least one non-missing post-baseline measure. Imputation by last observation carried forward (LOCF) for post-baseline values

Score ranging from 0 to 100 with higher scores indicating less bodily pain

Outcome measures

Outcome measures
Measure
Pramipexole
n=157 Participants
4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase the dose to 0.25mg and to further increase or decrease the dose in steps to 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Placebo
n=152 Participants
4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Change From Baseline in Short Form-36 (SF-36) Dimension Bodily Pain After 26 Weeks
12 Scores on a scale
Interval 0.0 to 31.0
9 Scores on a scale
Interval -1.0 to 24.5

SECONDARY outcome

Timeframe: Baseline and 26 weeks

Population: Intent to treat analysis. Number of randomized patients with a baseline and at least one non-missing post-baseline measure. Imputation by last observation carried forward (LOCF) for post-baseline values

Score ranging from 0 to 100 with higher scores indicating better health status

Outcome measures

Outcome measures
Measure
Pramipexole
n=155 Participants
4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase the dose to 0.25mg and to further increase or decrease the dose in steps to 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Placebo
n=152 Participants
4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Change From Baseline in SF-36 Dimension General Health After 26 Weeks
0 Scores on a scale
Interval -5.0 to 10.0
0 Scores on a scale
Interval -5.0 to 10.0

SECONDARY outcome

Timeframe: Baseline and 26 weeks

Population: Intent to treat analysis. Number of randomized patients with a baseline and at least one non-missing post-baseline measure. Imputation by last observation carried forward (LOCF) for post-baseline values

Score ranging from 0 to 100 with higher scores indicating better mental health

Outcome measures

Outcome measures
Measure
Pramipexole
n=155 Participants
4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase the dose to 0.25mg and to further increase or decrease the dose in steps to 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Placebo
n=152 Participants
4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Change From Baseline in SF-36 Dimension Mental Health After 26 Weeks
5 Scores on a scale
Interval -5.0 to 15.0
5 Scores on a scale
Interval -5.0 to 10.0

SECONDARY outcome

Timeframe: Baseline and 26 weeks

Population: Intent to treat analysis. Number of randomized patients with a baseline and at least one non-missing post-baseline measure. Imputation by last observation carried forward (LOCF) for post-baseline values

Score ranging from 0 to 100 with higher scores indicating better physical functioning

Outcome measures

Outcome measures
Measure
Pramipexole
n=156 Participants
4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase the dose to 0.25mg and to further increase or decrease the dose in steps to 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Placebo
n=152 Participants
4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Change From Baseline in SF-36 Dimension Physical Functioning After 26 Weeks
0 Scores on a scale
Interval 0.0 to 10.0
0 Scores on a scale
Interval -5.0 to 10.0

SECONDARY outcome

Timeframe: Baseline and 26 weeks

Population: Intent to treat analysis. Number of randomized patients with a baseline and at least one non-missing post-baseline measure. Imputation by last observation carried forward (LOCF) for post-baseline values

Score ranging from 0 to 100 with higher scores indicating less limitations due to emotional problems

Outcome measures

Outcome measures
Measure
Pramipexole
n=156 Participants
4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase the dose to 0.25mg and to further increase or decrease the dose in steps to 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Placebo
n=152 Participants
4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Change From Baseline in SF-36 Dimension Role Limitations Due to Emotional Problems After 26 Weeks
0 Scores on a scale
Interval -8.3 to 16.7
0 Scores on a scale
Interval 0.0 to 16.7

SECONDARY outcome

Timeframe: Baseline and 26 weeks

Population: Intent to treat analysis. Number of randomized patients with a baseline and at least one non-missing post-baseline measure. Imputation by last observation carried forward (LOCF) for post-baseline values

Score ranging from 0 to 100 with higher scores indicating less limitations due to physical problems

Outcome measures

Outcome measures
Measure
Pramipexole
n=156 Participants
4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase the dose to 0.25mg and to further increase or decrease the dose in steps to 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Placebo
n=152 Participants
4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Change From Baseline in SF-36 Dimension Role Limitations Due to Physical Problems After 26 Weeks
6.3 Scores on a scale
Interval 0.0 to 18.8
6.3 Scores on a scale
Interval 0.0 to 18.8

SECONDARY outcome

Timeframe: Baseline and 26 weeks

Population: Intent to treat analysis. Number of randomized patients with a baseline and at least one non-missing post-baseline measure. Imputation by last observation carried forward (LOCF) for post-baseline values

Score ranging from 0 to 100 with higher scores indicating better social functioning

Outcome measures

Outcome measures
Measure
Pramipexole
n=157 Participants
4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase the dose to 0.25mg and to further increase or decrease the dose in steps to 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Placebo
n=152 Participants
4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Change From Baseline in SF-36 Dimension Social Functioning After 26 Weeks
0 Scores on a scale
Interval 0.0 to 12.5
0 Scores on a scale
Interval 0.0 to 25.0

SECONDARY outcome

Timeframe: Baseline and 26 weeks

Population: Intent to treat analysis. Number of randomized patients with a baseline and at least one non-missing post-baseline measure. Imputation by last observation carried forward (LOCF) for post-baseline values

Score ranging from 0 to 100 with higher scores indicating better vitality

Outcome measures

Outcome measures
Measure
Pramipexole
n=155 Participants
4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase the dose to 0.25mg and to further increase or decrease the dose in steps to 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Placebo
n=152 Participants
4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Change From Baseline in SF-36 Dimension Vitality After 26 Weeks
6.3 Scores on a scale
Interval 0.0 to 18.8
3.1 Scores on a scale
Interval -6.3 to 12.5

SECONDARY outcome

Timeframe: Baseline and 26 weeks

Population: Intent to treat analysis. Number of randomized patients with a baseline and at least one non-missing post-baseline measure. Imputation by last observation carried forward (LOCF) for post-baseline values

Score ranging from 0 to 100 with higher scores indicating better health

Outcome measures

Outcome measures
Measure
Pramipexole
n=155 Participants
4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase the dose to 0.25mg and to further increase or decrease the dose in steps to 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Placebo
n=152 Participants
4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Change From Baseline in SF-36 Dimension Mental Component Summary After 26 Weeks
1.7 Scores on a scale
Interval -2.4 to 8.3
1.9 Scores on a scale
Interval -2.3 to 6.7

SECONDARY outcome

Timeframe: Baseline and 26 weeks

Population: Intent to treat analysis. Number of randomized patients with a baseline and at least one non-missing post-baseline measure. Imputation by last observation carried forward (LOCF) for post-baseline values

Score ranging from 0 to 100 with higher scores indicating better health

Outcome measures

Outcome measures
Measure
Pramipexole
n=155 Participants
4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase the dose to 0.25mg and to further increase or decrease the dose in steps to 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Placebo
n=152 Participants
4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Change From Baseline in SF-36 Dimension Physical Component Summary After 26 Weeks
2.1 Scores on a scale
Interval -0.5 to 7.5
2 Scores on a scale
Interval -2.0 to 5.9

SECONDARY outcome

Timeframe: after at least 4 weeks of treatment

Population: Treated Set and where patients received study medication for at least 4 weeks (Treated Set includes all patients who were documented to have taken at least one dose of of treatment)

Augmentation is a worsening of RLS symptoms and may manifest as increased severity and the involvement of other extremities or as a shift of RLS symptoms to a time period that is 2 or more hours earlier than was typical of the time of symptom onset during the initial course of beneficial stable treatment or the state before recently starting treatment.

Outcome measures

Outcome measures
Measure
Pramipexole
n=152 Participants
4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase the dose to 0.25mg and to further increase or decrease the dose in steps to 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Placebo
n=149 Participants
4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Diagnosis of Classified Augmentation According to Independent Expert Panel
18 participants
14 participants

SECONDARY outcome

Timeframe: after at least 1 week of treatment discontinuation

Population: Treated Set, all patients who were documented to have taken at least one dose of study medication

Worsening of RLS symptoms, in comparison to baseline, following abrupt treatment discontinuation (for patients with no added RLS therapy after study drug discontinuation). Assessment of worsening of RLS was based on the IRLS total score assessed 7 ± 1 days after treatment discontinuation (the end of the study or premature discontinuation) compared with that at baseline. Analysis considered the number of patients experiencing a clinically relevant deterioration of ≥4 points in total IRLS score 7 ± 1 days after discontinuation of trial medication compared with baseline.

Outcome measures

Outcome measures
Measure
Pramipexole
n=135 Participants
4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase the dose to 0.25mg and to further increase or decrease the dose in steps to 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Placebo
n=133 Participants
4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Worsening of RLS Symptoms (by at Least 4 Points in the IRLS Total Score Compared to Baseline) After Treatment Discontinuation
14 participants
2 participants

SECONDARY outcome

Timeframe: Baseline, Week 26

Population: Treated Set, all patients who were documented to have taken at least one dose of study medication

Outcome measures

Outcome measures
Measure
Pramipexole
n=166 Participants
4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase the dose to 0.25mg and to further increase or decrease the dose in steps to 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Placebo
n=163 Participants
4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Baseline, Week 26 Mean Supine Systolic Blood Pressure
Baseline
133.4 mm Hg
Standard Deviation 16.9
132.7 mm Hg
Standard Deviation 18.4
Baseline, Week 26 Mean Supine Systolic Blood Pressure
Week 26
132.3 mm Hg
Standard Deviation 16.4
132.2 mm Hg
Standard Deviation 16.5

SECONDARY outcome

Timeframe: Baseline, Week 26

Population: Treated Set, all patients who were documented to have taken at least one dose of study medication

Outcome measures

Outcome measures
Measure
Pramipexole
n=166 Participants
4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase the dose to 0.25mg and to further increase or decrease the dose in steps to 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Placebo
n=163 Participants
4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Baseline, Week 26 Mean Standing Systolic Blood Pressure
Baseline
132.6 mm Hg
Standard Deviation 17.3
130.6 mm Hg
Standard Deviation 18.2
Baseline, Week 26 Mean Standing Systolic Blood Pressure
Week 26
132.4 mm Hg
Standard Deviation 18.2
130.1 mm Hg
Standard Deviation 17.1

SECONDARY outcome

Timeframe: Baseline, Week 26

Population: Treated Set, all patients who were documented to have taken at least one dose of study medication

Outcome measures

Outcome measures
Measure
Pramipexole
n=166 Participants
4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase the dose to 0.25mg and to further increase or decrease the dose in steps to 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Placebo
n=163 Participants
4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Baseline, Week 26 Mean Supine Diastolic Blood Pressure
Baseline
79.2 mm Hg
Standard Deviation 9.7
79.6 mm Hg
Standard Deviation 9.7
Baseline, Week 26 Mean Supine Diastolic Blood Pressure
Week 26
78.3 mm Hg
Standard Deviation 9.7
79.5 mm Hg
Standard Deviation 9.4

SECONDARY outcome

Timeframe: Baseline, Week 26

Population: Treated Set, all patients who were documented to have taken at least one dose of study medication

Outcome measures

Outcome measures
Measure
Pramipexole
n=166 Participants
4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase the dose to 0.25mg and to further increase or decrease the dose in steps to 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Placebo
n=163 Participants
4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Baseline, Week 26 Mean Standing Diastolic Blood Pressure
Baseline
82.7 mm Hg
Standard Deviation 10.5
81.7 mm Hg
Standard Deviation 10.7
Baseline, Week 26 Mean Standing Diastolic Blood Pressure
Week 26
80.5 mm Hg
Standard Deviation 10.6
80.8 mm Hg
Standard Deviation 10.0

SECONDARY outcome

Timeframe: Baseline, Week 26

Population: Treated Set, all patients who were documented to have taken at least one dose of study medication

Outcome measures

Outcome measures
Measure
Pramipexole
n=166 Participants
4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase the dose to 0.25mg and to further increase or decrease the dose in steps to 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Placebo
n=163 Participants
4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Baseline, Week 26 Mean Supine Pulse Rate
Baseline
68.5 bpm
Standard Deviation 9.6
68.7 bpm
Standard Deviation 10.6
Baseline, Week 26 Mean Supine Pulse Rate
Week 26
69.1 bpm
Standard Deviation 8.9
68.3 bpm
Standard Deviation 10.6

SECONDARY outcome

Timeframe: Baseline, Week 26

Population: Treated Set, all patients who were documented to have taken at least one dose of study medication

Outcome measures

Outcome measures
Measure
Pramipexole
n=166 Participants
4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase the dose to 0.25mg and to further increase or decrease the dose in steps to 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Placebo
n=163 Participants
4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Baseline, Week 26 Mean Standing Pulse Rate
Baseline
74.6 bpm
Standard Deviation 10.2
74.0 bpm
Standard Deviation 10.7
Baseline, Week 26 Mean Standing Pulse Rate
Week 26
74.1 bpm
Standard Deviation 8.9
75.0 bpm
Standard Deviation 10.6

Adverse Events

Pramipexole

Serious events: 8 serious events
Other events: 70 other events
Deaths: 0 deaths

Placebo

Serious events: 3 serious events
Other events: 58 other events
Deaths: 0 deaths

Serious adverse events

Serious adverse events
Measure
Pramipexole
n=166 participants at risk
4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase the dose to 0.25mg and to further increase or decrease the dose in steps to 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Placebo
n=163 participants at risk
4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Infections and infestations
Appendicitis
0.00%
0/166 • 26 weeks
0.61%
1/163 • 26 weeks
Infections and infestations
Urinary tract infection
0.60%
1/166 • 26 weeks
0.00%
0/163 • 26 weeks
Infections and infestations
Viral infection
0.00%
0/166 • 26 weeks
0.61%
1/163 • 26 weeks
Cardiac disorders
Myocardial infarction
0.60%
1/166 • 26 weeks
0.00%
0/163 • 26 weeks
Vascular disorders
Orthostatic hypotension
0.00%
0/166 • 26 weeks
0.61%
1/163 • 26 weeks
Respiratory, thoracic and mediastinal disorders
Chronic obstructive pulmonary disease
0.60%
1/166 • 26 weeks
0.00%
0/163 • 26 weeks
Gastrointestinal disorders
Crohn's disease
0.00%
0/166 • 26 weeks
0.61%
1/163 • 26 weeks
Gastrointestinal disorders
Haemorrhoidal haemorrhage
0.60%
1/166 • 26 weeks
0.00%
0/163 • 26 weeks
Gastrointestinal disorders
Vomiting
0.00%
0/166 • 26 weeks
0.61%
1/163 • 26 weeks
Musculoskeletal and connective tissue disorders
Intervertebral disc protrusion
0.60%
1/166 • 26 weeks
0.00%
0/163 • 26 weeks
Musculoskeletal and connective tissue disorders
Neck pain
0.60%
1/166 • 26 weeks
0.00%
0/163 • 26 weeks
Reproductive system and breast disorders
Uterine prolapse
0.60%
1/166 • 26 weeks
0.00%
0/163 • 26 weeks
Injury, poisoning and procedural complications
Extradural haematoma
0.60%
1/166 • 26 weeks
0.00%
0/163 • 26 weeks
Injury, poisoning and procedural complications
Humerus fracture
0.60%
1/166 • 26 weeks
0.00%
0/163 • 26 weeks

Other adverse events

Other adverse events
Measure
Pramipexole
n=166 participants at risk
4 weeks of flexible dose-titration (to optimise efficacy and tolerability), starting at 0.125 mg once daily with the potential to increase the dose to 0.25mg and to further increase or decrease the dose in steps to 0.5 mg and 0.75 mg, with the final dose level subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Placebo
n=163 participants at risk
4 weeks of flexible dose-titration as for the investigational product; with the dose subsequently fixed for 22 weeks. mode of administration: Oral, once daily in the evening (2 to 3 hours before bedtime) form: tablets
Gastrointestinal disorders
Nausea
14.5%
24/166 • 26 weeks
3.7%
6/163 • 26 weeks
General disorders
Fatigue
10.8%
18/166 • 26 weeks
9.2%
15/163 • 26 weeks
Nervous system disorders
Headache
7.8%
13/166 • 26 weeks
10.4%
17/163 • 26 weeks
Nervous system disorders
Restless legs syndrome
6.6%
11/166 • 26 weeks
6.7%
11/163 • 26 weeks
Nervous system disorders
Somnolence
6.6%
11/166 • 26 weeks
4.9%
8/163 • 26 weeks
Infections and infestations
Nasopharyngitis
4.2%
7/166 • 26 weeks
6.1%
10/163 • 26 weeks
Musculoskeletal and connective tissue disorders
Muscle spasms
6.0%
10/166 • 26 weeks
2.5%
4/163 • 26 weeks
Musculoskeletal and connective tissue disorders
Arthralgia
5.4%
9/166 • 26 weeks
1.2%
2/163 • 26 weeks

Additional Information

Boehringer Ingelheim Call Center

Boehringer Ingelheim Pharmaceuticals

Phone: 1-800-243-0127

Results disclosure agreements

  • Principal investigator is a sponsor employee Any publication of the result of this trial must be consistent with the Boehringer Ingelheim publication policy. The rights of the investigator and of the sponsor with regard to publication of the results of this trial are described in the investigator contract.
  • Publication restrictions are in place

Restriction type: OTHER